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Src kinase
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Curated Studies
Most Correlated Studies
Mammary gland epithelial MCF 10A cells overexpressing tyrosine-protein kinase SRC
Ovarian tumor biopsies from a Phase I dasatinib trial
Clear cell carcinoma of kidney ACHN cells treated with Dasatinib and Cabozantinib
Glioblastoma LN229 cells treated with UM-164
Embryonic fibroblasts and neuroretinal cells transformed with Rous sarcoma virus
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Literature
Most Relevant Literature
CSK-homologous kinase (CHK/MATK) is a potential colorectal cancer tumour suppressor gene epigenetica…
Csk αC Helix: A Computational Analysis of an Essential Region for Conformational Transitions.
SH3-domain mutations selectively disrupt Csk homodimerization or PTPN22 binding.
Acute Csk inhibition hinders B cell activation by constraining the PI3 kinase pathway.
Inhibiting ACK1-mediated phosphorylation of C-terminal Src kinase counteracts prostate cancer immune…
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Clinical Trials
Most Relevant Clinical Trials
PH I SRC Kinase, Dasatinib Combo Paclitaxel & Carboplatin in Pts w Ovarian, Peritoneal, & Tubal Canc…
Insulin-like Growth Factor 1 Receptor (IGF-1R) Antibody AMG479 (Ganitumab) in Combination With the S…
Bristol-Myers Squibb Dasatinib Src Inhibition in Endometrial Cancer
Comparison of Biomarker Modulation by Inhibition of EGFR and/or SRC Family
SRC Inhibition as a Potential Target for Parkinson's Disease Psychosis
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