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mat2a protein, human
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Development of a Series of Pyrrolopyridone MAT2A Inhibitors.
Discovery of novel MAT2A inhibitors by an allosteric site-compatible fragment growing approach.
Discovery of novel methionine adenosyltransferase 2A (MAT2A) allosteric inhibitors by structure-base…
Identification of a Sonically Activated Degrader of Methionine Adenosyltransferase 2A by an in Silic…
Blocking methionine catabolism induces senescence and confers vulnerability to GSK3 inhibition in li…
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AMG 193, Methylthioadenosine (MTA) Cooperative Protein Arginine Methyltransferase 5 (PRMT5) Inhibito…
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