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cyclin-dependent protein serine/threonine kinase inhibitor activity
(biogroup)
Summary
General Info
Body Atlas
Most Correlated Tissues
Vagina
Stomach
Skeletal muscle
Testes
Salivary gland
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Disease Atlas
Most Correlated Diseases
Vesicular stomatitis Indiana virus disease
Myocardial ischemia
Perforation of tympanic membrane
Infection due to Mycobacterium tuberculosis
Injury of integument
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Pharmaco Atlas
Most Correlated Compounds
Apitolisib
RPI-1 cpd
((3Z)-N-(3-chlorophenyl)-3-((3,5-dimethyl-4-((4-methylpiperazin-1-yl)carbonyl)-1H-pyrrol-2-yl)methylene)-N-methyl-2-oxo-2,3-dihydro-1H-indole-5-sulfonamide)
SB 525334
ompP2 protein, Haemophilus influenzae
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Knockdown Atlas
Most Correlated Gene Perturbations
CASP8AP2
ZBTB16
BAK1
NR5A1
ZCCHC24
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Curated Studies
Most Correlated Studies
Oral keratinocytes HOK16B cells treated with cannabidiol before LPS + ATP mediated inflammation
Gene expression from U937T:PLZF-RARa Inducible Cells
L1000 CMAP - Colorectal cancer HT29.311 cells with CRISPR-targeted gene knockouts
HCT116 cells isogenic for p53 expression upon treatment with actinomycin D and nutlin-3
L1000 CMAP - Breast cancer MCF7 cells treated with small molecule perturbagens (1 of 4)
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Literature
Most Relevant Literature
Identification of novel molecular markers through transcriptomic analysis in human fetal and adult c…
Melatonin-induced gene expression changes and its preventive effects on adriamycin-induced lipid per…
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Clinical Trials
Most Relevant Clinical Trials
A Phase II Window of Opportunity Trial of PRMT5 Inhibitor, GSK3326595, in Early Stage Breast Cancer
A Study of Palbociclib in Addition to Standard Endocrine Treatment in Hormone Receptor Positive Her2…
Study Of Real-World Evidence In Patients Treated With Palbociclib During a 2.5 Years Follow-Up Perio…
Dose Escalation and Expansion Study of GSK525762 in Combination With Fulvestrant in Subjects With Ho…
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